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- A4130 ENMD-2076Target: Aurora Kinases|FLT3|RET|Src|VEGFR3/FLT4|NTRK1/TRKA|CSF-1R/c-FmsSummary: Aurora A/Flt3的选择性抑制剂
- A2187 Cladribine中文名: 克拉利宾Target: Adenosine DeaminasesSummary: 白血病细胞凋亡诱导物
- A3708 Pentostatin1 Citation中文名: 喷司他丁Target: Adenosine DeaminasesSummary: 腺苷脱氨酶抑制剂
- A2571 Pepstatin A1 Citation中文名: 抑肽素Target: Cathepsins|Renin|HIV proteases|PepsinsSummary: 天冬氨酸蛋白酶抑制剂