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- A8171 Entinostat (MS-275,SNDX-275)2 Citation中文名: 恩替诺特Target: Histone Deacetylases (HDACs)Summary: HDAC1和HDAC3抑制剂
- A3603 MI-3Target: Menin-MLLSummary: Menin-MLL抑制剂
- A8317 Fludarabine Phosphate (Fludara)2 Citation中文名: 磷酸氟达拉滨Target: STATSummary: 抑制STAT1激活和DNA合成
- B3283 PF-04449913中文名: 格拉吉布Target: SmoothenedSummary: Smoothened拮抗剂
- B2114 Mitoxantrone HCl中文名: 米托蒽醌Target: Pim|Topoisomerases|USP|HIV IntegrasesSummary: 拓扑异构酶II抑制剂
- A4139 AG-4903 CitationTarget: EGFR|JAKSummary: JAK2/EGFR抑制剂
- A4138 Tofacitinib (CP-690550,Tasocitinib)1 Citation中文名: 托法替尼,托法替布Target: JAKSummary: Janus激酶抑制剂
- A8341 Go 6976Target: PKCSummary: PKC α/PKC β1抑制剂
- A4148 NVP-BSK805 2HClTarget: JAKSummary: JAK2抑制剂
- B1250 Ezatiostat hydrochloride3 CitationTarget: Gutathione S-transferaseSummary: GST抑制剂