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- A3962 AZD1208Target: PimSummary: PIM激酶抑制剂
- A3556 LKB1 (AAK1 dual inhibitor)Target: PimSummary: Pim-1激酶抑制剂
- A4130 ENMD-2076Target: Aurora Kinases|FLT3|RET|Src|VEGFR3/FLT4|NTRK1/TRKA|CSF-1R/c-FmsSummary: Aurora A/Flt3的选择性抑制剂
- N1842 Taxifolin中文名: 紫杉叶素,黄杉素Target: AdipoR2|Opioid receptors
- A8236 Regorafenib4 Citation中文名: 瑞戈非尼Target: Raf|VEGFR|PDGFR|c-Kit|RETSummary: VEGFR/PDGFR/FGFR/mutant Kit/RET/Raf-1抑制剂