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- A3018 Trametinib (GSK1120212)7 Citation中文名: 曲美替尼Target: MEKSummary: MEK1和MEK2抑制剂
- A3394 Epothilone D中文名: 埃博霉素 DTarget: Microtubule/TubulinSummary: 天然聚酮化合物
- A3887 Trametinib DMSO solvate1 CitationTarget: MEKSummary: 变构MEK1/MEK2 激酶抑制剂
- A1947 MEK162 (ARRY-162, ARRY-438162)中文名: 贝美替尼Target: MEKSummary: MEK1/2抑制剂
- A5573 Pimasertib (AS-703026)Target: MEKSummary: MEK1/2抑制剂