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- N2135 Gossypol2 Citation中文名: 棉籽酚,棉酚Target: DehydrogenaseSummary: PAF抑制剂,抗生育和抗癌
- B1317 ML-323Target: Deubiquitinating enzymes (DUBs)Summary: USP1-UAF1抑制剂
- A8212 PR-619Target: Deubiquitinating enzymes (DUBs)Summary: 去泛素化酶(DUBs)抑制剂
- A8340 Cyclopamine1 Citation中文名: 环巴胺Target: SmoothenedSummary: Hedgehog (Hh)信号抑制剂
- A5703 BMS-777607Target: METSummary: 强效的c-Met选择性抑制剂