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- A3927 VS-5584 (SB2343)Target: PI3K|mTORSummary: MTOR/P13K抑制剂
- A4390 Pemetrexed1 Citation中文名: 培美曲塞二钠盐Target: Thymidylate Synthase|DHFR|GARFTSummary: TS、DHFR、GARFT和AICARFT抑制剂
- A4203 Tenovin-1Target: Sir2-like Family Deacetylases (Sirtuins)|p53|p21Summary: SIRT2 抑制剂,p53激活剂
- A8169 Everolimus (RAD001)8 Citation中文名: 依维莫司Target: mTORSummary: MTOR抑制剂
- A5078 KU-0063794Target: mTORSummary: mTORC1和mTORC2的抑制剂
- A8394 CHIR-124Target: FLT3|GSK-3|Chk|PDGFRSummary: Chk1抑制剂
- A8312 Torin 17 CitationTarget: mTORSummary: MTOR抑制剂
- A8477 MK-8776 (SCH-900776)Target: ChkSummary: Chk1高效选择性抑制剂