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- A2942 Masitinib (AB1010)中文名: 马赛替尼Target: PDGFR|c-Kit|LynSummary: 酪氨酸激酶抑制剂
- A8539 Tretinoin (Aberela)中文名: 维A酸Target: RAR/RXRSummary: 视黄酸,用于治疗痤疮和毛发角化病.
- B1317 ML-323Target: Deubiquitinating enzymes (DUBs)Summary: USP1-UAF1抑制剂
- A8212 PR-619Target: Deubiquitinating enzymes (DUBs)Summary: 去泛素化酶(DUBs)抑制剂
- A5703 BMS-777607Target: METSummary: 强效的c-Met选择性抑制剂