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- A2942 Masitinib (AB1010)中文名: 马赛替尼Target: PDGFR|c-Kit|LynSummary: 酪氨酸激酶抑制剂
- A3732 PoloxinTarget: PLKSummary: PLK1抑制剂
- A3962 AZD1208Target: PimSummary: PIM激酶抑制剂
- A4122 PHA-680632Target: Aurora Kinases|PLK|FGFRSummary: Aurora激酶抑制剂
- A5979 Tie2 kinase inhibitor中文名: Tie2激酶抑制剂Target: Tie-2Summary: Tie-2(Tie2 )抑制剂