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- A3927 VS-5584 (SB2343)Target: PI3K|mTORSummary: MTOR/P13K抑制剂
- A5072 GSK690693Target: Akt|PKC|PKG|PKA|PrkSummary: ATP竞争性的Pan-AKT抑制剂
- A5057 MGCD-265Target: VEGFR|c-METSummary: Met/Flt/Flk/Ron/Tie-2抑制剂
- A2942 Masitinib (AB1010)中文名: 马赛替尼Target: PDGFR|c-Kit|LynSummary: 酪氨酸激酶抑制剂
- A3732 PoloxinTarget: PLKSummary: PLK1抑制剂
- A3433 Gefitinib hydrochloride中文名: 盐酸吉非替尼Target: EGFRSummary: EGFR有效的抑制剂
- A8327 Verteporfin中文名: 维替泊芬Target: YAPSummary: 光增敏剂
- A8446 Ibuprofen中文名: 布洛芬Target: COXSummary: 生物学活性
- A8539 Tretinoin (Aberela)中文名: 维A酸Target: RAR/RXRSummary: 视黄酸,用于治疗痤疮和毛发角化病.
- A8178 Panobinostat (LBH589)10 Citation中文名: 帕比司他Target: Histone Deacetylases (HDACs)Summary: HDAC抑制剂