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- A3005 CAL-101 (Idelalisib, GS-1101)2 Citation中文名: 艾代拉里斯,艾代拉利司Target: PI3KSummary: PI3K抑制剂
- A4482 Pifithrin-μ1 CitationTarget: Autophagy|p53|HSP70Summary: p53结合抑制剂,抗凋亡。
- A3214 AZD11521 CitationTarget: Aurora KinasesSummary: Aurora B激酶抑制剂
- A4124 TAK-901Target: Aurora Kinases|FLT3|Src|JAK|LRRK2|Hck|FGR|YES|Fyn|ARGSummary: Aurora A/B抑制剂
- A4121 SNS-314 MesylateTarget: Aurora KinasesSummary: Aurora A/B/C激酶抑制剂
- B1047 GDC-0032Target: PI3KSummary: PI3Kα 抑制剂
- A4116 Danusertib (PHA-739358)2 Citation中文名: 达鲁舍替Target: Aurora KinasesSummary: Aurora kinase(极光激酶)抑制剂