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- A8236 Regorafenib4 Citation中文名: 瑞戈非尼Target: Raf|VEGFR|PDGFR|c-Kit|RETSummary: VEGFR/PDGFR/FGFR/mutant Kit/RET/Raf-1抑制剂
- B7782 BRD 7552Target: Pancreatic and duodenal homeobox 1 (PDX1)Summary: PDX1诱导剂
- A1630 Epothilone B (EPO906, Patupilone)中文名: 埃博霉素B,帕土匹龙Target: Microtubules/TubulinsSummary: 大环内酯物抗癌试剂
- A3183 Ansamitocin P-3中文名: 安丝菌素 P 3'Target: Microtubules/TubulinsSummary: 美登素类似物,微管蛋白抑制剂
- B5835 AZD2932Target: FLT3|VEGFR|PDGFR|c-KitSummary: VEGFR-2\PDGFRβ\Flt-3和c-Kit的抑制剂
- A4213 Necrostatin-15 CitationTarget: RIP kinasesSummary: RIP1抑制剂