Signaling Pathways - Flk1 - DGAT - DREADD Ligands - Thymidylate Synthase - Carbonic Anhydrases
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- B3709 Midostaurin (PKC412)中文名: 米哚妥林Target: PKC|PKA|KDR|Flk1|PPK|c-Syk|CDK1/CyclinBSummary: PKC抑制剂
- B1476 Raltitrexed中文名: 雷替曲塞Target: Thymidylate SynthaseSummary: 胸苷酸合酶抑制剂
- B1279 Dorzolamide中文名: 多佐胺Target: Carbonic AnhydrasesSummary: 碳酸酐酶抑制剂
- A8397 Chlorothiazide中文名: 氯噻嗪Target: Carbonic AnhydrasesSummary: 碳酸酐酶抑制剂
- A8473 Methyocarbamol中文名: 美索巴莫Target: Carbonic AnhydrasesSummary: 碳酸酐酶抑制剂
- A5354 Zonisamide中文名: 唑尼沙胺Target: Voltage-gated Sodium (NaV) Channels|Voltage-gated Calcium Channels (CaV)|Carbonic Anhydrases|Calcium-Activated Potassium (KCa) ChannelsSummary: 抗惊厥和机械效应的抗癫痫药
- A2597 Brivanib (BMS-540215)中文名: 布立尼布Target: VEGFR|FGFR|Flk1Summary: VEGFR-2的ATP竞争性抑制剂
- A3317 Clozapine N-oxide(CNO)1 Citation中文名: 氯氮平的N-氧化物Target: DREADD LigandsSummary: Clozapine代谢产物,用于化学遗传学
- A3215 AZD7687Target: DGATSummary: 强效的选择性DGAT抑制剂
- A4390 Pemetrexed1 Citation中文名: 培美曲塞二钠盐Target: Thymidylate Synthase|DHFR|GARFTSummary: TS、DHFR、GARFT和AICARFT抑制剂