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Signaling Pathways - sodium channel - Phosphodiesterases (PDEs)

19件产品中的 1-10

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  1. BRL 50481
    B6988 BRL 50481
    Target: Phosphodiesterases (PDEs)
    Summary: PDE7抑制剂
      Soluble in DMSO
  2. Etazolate hydrochloride
    B6304 Etazolate hydrochloride
     2 Citation
    Target: Phosphodiesterases (PDEs)
    Summary: PDE-4抑制剂和选择性GABA-A受体调节剂
      ≥7.75 mg/mL
      insoluble in H2O
  3. Udenafil
    B3439 Udenafil
    中文名: 乌地那非
    Target: Phosphodiesterases (PDEs)
    Summary: PDE5抑制剂
      ≥117.2 mg/mL
      insoluble in H2O
  4. Ibutilide Fumarate
    B2278 Ibutilide Fumarate
    中文名: 富马酸伊布利特
    Target: Voltage-gated Potassium (KV) Channels|Voltage-gated Calcium Channels (CaV)|sodium channel
    Summary: III类抗心律失常药物
      ≥25.6 mg/mL
      ≥16.4 mg/mL
  5. Lamotrigine
    B2249 Lamotrigine
     1 Citation
    中文名: 拉莫三嗪
    Target: 5-HT receptors|sodium channel
    Summary: 5-HT抑制剂,钠通道阻断剂
      ≥12.3 mg/mL
      insoluble in H2O
  6. Milrinone
    B1386 Milrinone
    中文名: 米力农
    Target: Phosphodiesterases (PDEs)
    Summary: PDE3抑制剂
      ≥8.2 mg/mL
      insoluble in H2O
  7. Vinpocetine
    B2276 Vinpocetine
    中文名: 长春西汀
    Target: Phosphodiesterases (PDEs)
    Summary: PDE抑制剂
      ≥5.83 mg/mL
      ≥2.59 mg/mL
  8. Dronedarone
    A3374 Dronedarone
    中文名: 决奈达隆
    Target: Cytochrome P450 (CYP450)|sodium channel|adrenergic receptor|potassium channel|calcium channel
    Summary: CYP3A4和2D6抑制剂
      ≥27.84 mg/mL
      insoluble in H2O
  9. Deltarasin
    A3358 Deltarasin
    Target: Phosphodiesterases (PDEs)
    Summary: KRAS-PDEδ相互作用抑制剂
      Soluble in DMSO
  10. Aminophylline
    A4346 Aminophylline
    中文名: 氨茶碱,氨基非林
    Target: Phosphodiesterases (PDEs)
    Summary: Pan-PDE抑制剂
      ≥13.48 mg/mL
      ≥14.45 mg/mL

19件产品中的 1-10

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