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Signaling Pathways - KDM - sodium channel - CysLT1 - Phosphodiesterases (PDEs)

22件产品中的 1-10

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  1. TC-E 5002
    B4930 TC-E 5002
    Target: KDM
    Summary: 选择性组蛋白去甲基化酶KDM2/7亚家族抑制剂
      Soluble in DMSO
  2. MK-571 sodium salt hydrate
    B8031 MK-571 sodium salt hydrate
     3 Citation
    Target: CysLT1
    Summary: CysLT1受体拮抗剂
      ≥10.3 mg/mL
      ≥122.2 mg/mL
  3. BRL 50481
    B6988 BRL 50481
    Target: Phosphodiesterases (PDEs)
    Summary: PDE7抑制剂
      Soluble in DMSO
  4. Etazolate hydrochloride
    B6304 Etazolate hydrochloride
     2 Citation
    Target: Phosphodiesterases (PDEs)
    Summary: PDE-4抑制剂和选择性GABA-A受体调节剂
      ≥7.75 mg/mL
      insoluble in H2O
  5. Udenafil
    B3439 Udenafil
    中文名: 乌地那非
    Target: Phosphodiesterases (PDEs)
    Summary: PDE5抑制剂
      ≥117.2 mg/mL
      insoluble in H2O
  6. Ibutilide Fumarate
    B2278 Ibutilide Fumarate
    中文名: 富马酸伊布利特
    Target: Voltage-gated Potassium (KV) Channels|Voltage-gated Calcium Channels (CaV)|sodium channel
    Summary: III类抗心律失常药物
      ≥25.6 mg/mL
      ≥16.4 mg/mL
  7. Lamotrigine
    B2249 Lamotrigine
     1 Citation
    中文名: 拉莫三嗪
    Target: 5-HT receptors|sodium channel
    Summary: 5-HT抑制剂,钠通道阻断剂
      ≥12.3 mg/mL
      insoluble in H2O
  8. Milrinone
    B1386 Milrinone
    中文名: 米力农
    Target: Phosphodiesterases (PDEs)
    Summary: PDE3抑制剂
      ≥8.2 mg/mL
      insoluble in H2O
  9. Vinpocetine
    B2276 Vinpocetine
    中文名: 长春西汀
    Target: Phosphodiesterases (PDEs)
    Summary: PDE抑制剂
      ≥5.83 mg/mL
      ≥2.59 mg/mL
  10. Dronedarone
    A3374 Dronedarone
    中文名: 决奈达隆
    Target: Cytochrome P450 (CYP450)|sodium channel|adrenergic receptor|potassium channel|calcium channel
    Summary: CYP3A4和2D6抑制剂
      ≥27.84 mg/mL
      insoluble in H2O

22件产品中的 1-10

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