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Signaling Pathways - KDM - sodium channel - Hypoxia Inducible Factors (HIFs) - Calcium-Activated Potassium (KCa) Channels

10 件产品

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  1. PX-478 2HCl
    B6004 PX-478 2HCl
    Target: Hypoxia Inducible Factors (HIFs)
    Summary: HIF-1α抑制剂
      ≥19.7 mg/mL
      ≥50 mg/mL
  2. TC-E 5002
    B4930 TC-E 5002
    Target: KDM
    Summary: 选择性组蛋白去甲基化酶KDM2/7亚家族抑制剂
      Soluble in DMSO
  3. Ibutilide Fumarate
    B2278 Ibutilide Fumarate
    中文名: 富马酸伊布利特
    Target: Voltage-gated Potassium (KV) Channels|Voltage-gated Calcium Channels (CaV)|sodium channel
    Summary: III类抗心律失常药物
      ≥25.6 mg/mL
      ≥16.4 mg/mL
  4. Lamotrigine
    B2249 Lamotrigine
     1 Citation
    中文名: 拉莫三嗪
    Target: 5-HT receptors|sodium channel
    Summary: 5-HT抑制剂,钠通道阻断剂
      ≥12.3 mg/mL
      insoluble in H2O
  5. Dequalinium Chloride
    B2191 Dequalinium Chloride
    中文名: 地喹氯铵
    Target: PKC|Calcium-Activated Potassium (KCa) Channels
    Summary: PKC抑制剂
      insoluble in DMSO
      insoluble in H2O
  6. BAY 87-2243
    B1115 BAY 87-2243
    Target: Hypoxia Inducible Factors (HIFs)
    Summary: 有效的HIF-1选择性抑制剂
      ≥8.76 mg/mL
      insoluble in H2O
  7. Zonisamide
    A5354 Zonisamide
    中文名: 唑尼沙胺
    Target: Voltage-gated Sodium (NaV) Channels|Voltage-gated Calcium Channels (CaV)|Carbonic Anhydrases|Calcium-Activated Potassium (KCa) Channels
    Summary: 抗惊厥和机械效应的抗癫痫药
      ≥8.35 mg/mL
      insoluble in H2O
  8. TRAM-34
    A1888 TRAM-34
    Target: Calcium-Activated Potassium (KCa) Channels
    Summary: KCa3.1阻断剂
      ≥17.25 mg/mL
      insoluble in H2O
  9. Dronedarone
    A3374 Dronedarone
    中文名: 决奈达隆
    Target: Cytochrome P450 (CYP450)|sodium channel|adrenergic receptor|potassium channel|calcium channel
    Summary: CYP3A4和2D6抑制剂
      ≥27.84 mg/mL
      insoluble in H2O
  10. Daminozide
    A3348 Daminozide
    中文名: 丁酰肼
    Target: KDM|PHF
    Summary: KDM2A抑制剂
      ≥7.3 mg/mL
      ≥21.4 mg/mL

10 件产品

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