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Signaling Pathways - ETA Receptors - Bcl-xl - nuclear export - adrenergic receptor

10 件产品

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  1. IRL-2500
    B6872 IRL-2500
    Target: ETA Receptors|ETB Receptors
    Summary: 内皮素受体拮抗剂
  2. Epinephrine Bitartrate
    B1358 Epinephrine Bitartrate
    中文名: 酒石酸肾上腺素
    Target: adrenergic receptor
    Summary: 肾上腺素能受体激动剂
      ≥16.66 mg/mL
      ≥22.9 mg/mL
  3. Latrepirdine
    B1572 Latrepirdine
    Target: Voltage-gated Calcium Channels (CaV)|NMDA receptor|adrenergic receptor|Histamine receptors|GluR|5-HT receptor|dopamine receptors|AMPA receptor
    Summary: 脑细胞死亡抑制剂
      ≥19.62 mg/mL
      insoluble in H2O
  4. KPT-276
    B1463 KPT-276
    Target: nuclear export|CRM1
    Summary: CRM1抑制剂
      ≥19.85 mg/mL
      insoluble in H2O
  5. Ambrisentan
    B2075 Ambrisentan
    中文名: 安贝生坦
    Target: ETA Receptors
    Summary: ETA受体拮抗剂
      ≥18.92 mg/mL
      insoluble in H2O
  6. WEHI-539
    A3935 WEHI-539
     15 Citation
    Target: Bcl-xl
    Summary: 选择性的Bcl-xL抑制剂
      insoluble in DMSO
      insoluble in H2O
  7. Quetiapine
    A3744 Quetiapine
    中文名: 喹硫平
    Target: AChR|adrenergic receptor|5-HT receptor|Dopamine receptor|Histamine receptor
    Summary: 多巴胺受体拮抗剂
      ≥19.18 mg/mL
      insoluble in H2O
  8. Dronedarone
    A3374 Dronedarone
    中文名: 决奈达隆
    Target: Cytochrome P450 (CYP450)|sodium channel|adrenergic receptor|potassium channel|calcium channel
    Summary: CYP3A4和2D6抑制剂
      ≥27.84 mg/mL
      insoluble in H2O
  9. Apogossypolone (ApoG2)
    A4200 Apogossypolone (ApoG2)
     2 Citation
    Target: Bcl-2|Bcl-xl|Mcl-1
    Summary: Bcl-2的非肽类小分子抑制剂
      ≥24.55 mg/mL
      insoluble in H2O
  10. TW-37
    A4234 TW-37
     1 Citation
    Target: Bcl-2|Bcl-xl|Mcl-1
    Summary: Bcl-2抑制剂,抑制Bcl-2、Bcl-XL和Mcl-1。
      ≥19.75 mg/mL
      insoluble in H2O

10 件产品

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