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Signaling Pathways - DREADD Ligands - 5-HT3 Receptors - Flk1 - potassium channel

10 件产品

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  1. Midostaurin (PKC412)
    B3709 Midostaurin (PKC412)
    中文名: 米哚妥林
    Target: PKC|PKA|KDR|Flk1|PPK|c-Syk|CDK1/CyclinB
    Summary: PKC抑制剂
      ≥57.1 mg/mL
      insoluble in H2O
  2. Ondansetron
    B2241 Ondansetron
    中文名: 昂丹司琼
    Target: 5-HT3 Receptors
    Summary: 血清素5-HT3受体拮抗剂
      ≥7.33 mg/mL
      insoluble in H2O
  3. VUF 10166
    B2259 VUF 10166
    Target: 5-HT3 Receptors
    Summary: 5-HT3受体拮抗剂
      ≥38.8 mg/mL
      insoluble in H2O
  4. Tropisetron Hydrochloride
    B2258 Tropisetron Hydrochloride
    中文名: 盐酸托烷司琼
    Target: 5-HT3 Receptors
    Summary: 5-HT3受体拮抗剂
      ≥28.4 mg/mL
      ≥9.7 mg/mL
  5. Ondansetron HCl
    A5166 Ondansetron HCl
    中文名: 盐酸昂丹司琼
    Target: 5-HT3 Receptors
    Summary: 5-HT3受体拮抗剂
      ≥33.04 mg/mL
      insoluble in H2O
  6. Brivanib (BMS-540215)
    A2597 Brivanib (BMS-540215)
    中文名: 布立尼布
    Target: VEGFR|FGFR|Flk1
    Summary: VEGFR-2的ATP竞争性抑制剂
      ≥18.5 mg/mL
      insoluble in H2O
  7. Mosapride Citrate
    A1334 Mosapride Citrate
    中文名: 莫沙必利柠檬酸盐
    Target: 5-HT3 Receptors|5-HT4 Receptors
    Summary: 5-HT受体激动剂
      ≥30.7 mg/mL
      insoluble in H2O
  8. Vortioxetine
    A3926 Vortioxetine
    中文名: 沃替西汀
    Target: 5-HT1 Receptors|5-HT7 Receptors|5-HT3 Receptors|SERT
    Summary: 5-HT受体拮抗剂
      ≥14.92 mg/mL
      insoluble in H2O
  9. Dronedarone
    A3374 Dronedarone
    中文名: 决奈达隆
    Target: Cytochrome P450 (CYP450)|sodium channel|adrenergic receptor|potassium channel|calcium channel
    Summary: CYP3A4和2D6抑制剂
      ≥27.84 mg/mL
      insoluble in H2O
  10. Clozapine N-oxide(CNO)
    A3317 Clozapine N-oxide(CNO)
     1 Citation
    中文名: 氯氮平的N-氧化物
    Target: DREADD Ligands
    Summary: Clozapine代谢产物,用于化学遗传学
      ≥17.15 mg/mL
      ≥49 mg/mL

10 件产品

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