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Signaling Pathways - DREADD Ligands - SGLT - p53 - Voltage-gated Potassium (KV) Channels

15件产品中的 1-10

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  1. Psora 4
    B7659 Psora 4
     1 Citation
    Target: Voltage-gated Potassium (KV) Channels
    Summary: Kv1.3阻断剂
      ≥15.75 mg/mL
      insoluble in H2O
  2. Ibutilide Fumarate
    B2278 Ibutilide Fumarate
    中文名: 富马酸伊布利特
    Target: Voltage-gated Potassium (KV) Channels|Voltage-gated Calcium Channels (CaV)|sodium channel
    Summary: III类抗心律失常药物
      ≥25.6 mg/mL
      ≥16.4 mg/mL
  3. Cisapride
    B1198 Cisapride
    Target: Voltage-gated Potassium (KV) Channels|5-HT4 Receptor
    Summary: 5-HT4受体激动剂
      ≥23.3 mg/mL
      insoluble in H2O
  4. Terfenadine
    A8534 Terfenadine
    中文名: 特非那定
    Target: Voltage-gated Potassium (KV) Channels|Histamine H1 Receptors|Inward Rectifier Potassium (Kir) Channels
    Summary: 组胺H1受体拮抗剂
      ≥18 mg/mL
      insoluble in H2O
  5. Canagliflozin
    A8333 Canagliflozin
     1 Citation
    中文名: 卡格列净
    Target: SGLT
    Summary: SGLT2的有效选择性抑制剂
      ≥22.25 mg/mL
      insoluble in H2O
  6. Pifithrin-μ
    A4482 Pifithrin-μ
     1 Citation
    Target: Autophagy|p53|HSP70
    Summary: p53结合抑制剂,抗凋亡。
      ≥18.1 mg/mL
      insoluble in H2O
  7. PRIMA-1
    A4483 PRIMA-1
    Target: p53
    Summary: BAX抑制剂
      ≥9.1 mg/mL
      ≥110.6 mg/mL
  8. PhiKan 083
    A4481 PhiKan 083
    Target: p53
    Summary: P53稳定剂
      <27.48 mg/mL
      <13.74 mg/mL
  9. Phloretin
    A3723 Phloretin
    中文名: 根皮素
    Target: SGLT
    Summary: 在苹果中发现的二氢查耳酮
      ≥105 mg/mL
      insoluble in H2O
  10. Clozapine N-oxide(CNO)
    A3317 Clozapine N-oxide(CNO)
     1 Citation
    中文名: 氯氮平的N-氧化物
    Target: DREADD Ligands
    Summary: Clozapine代谢产物,用于化学遗传学
      ≥17.15 mg/mL
      ≥49 mg/mL

15件产品中的 1-10

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