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Signaling Pathways - Calcium-Activated Potassium (KCa) Channels - NAE - HCV polymerase - Glucagon-like peptide 1 (GLP-1) receptors

10 件产品

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  1. Exendin-3 (9-39) amide
    B6943 Exendin-3 (9-39) amide
     1 Citation
    Target: Glucagon-like peptide 1 (GLP-1) receptors
    Summary: GLP-1受体拮抗剂
      ≥168.5 mg/mL
      ≥25.2 mg/mL
  2. Dequalinium Chloride
    B2191 Dequalinium Chloride
    中文名: 地喹氯铵
    Target: PKC|Calcium-Activated Potassium (KCa) Channels
    Summary: PKC抑制剂
      insoluble in DMSO
      insoluble in H2O
  3. MLN4924
    B1036 MLN4924
     5 Citation
    Target: NAE|Ubiquitin-activating Enzyme E1|SUMOylation
    Summary: NAE抑制剂
      ≥22.18 mg/mL
      insoluble in H2O
  4. Zonisamide
    A5354 Zonisamide
    中文名: 唑尼沙胺
    Target: Voltage-gated Sodium (NaV) Channels|Voltage-gated Calcium Channels (CaV)|Carbonic Anhydrases|Calcium-Activated Potassium (KCa) Channels
    Summary: 抗惊厥和机械效应的抗癫痫药
      ≥8.35 mg/mL
      insoluble in H2O
  5. TRAM-34
    A1888 TRAM-34
    Target: Calcium-Activated Potassium (KCa) Channels
    Summary: KCa3.1阻断剂
      ≥17.25 mg/mL
      insoluble in H2O
  6. PSI-7977
    A3738 PSI-7977
    中文名: 索非布韦,索氟布韦
    Target: HCV polymerase
    Summary: 慢性丙型肝炎病毒(HCV)感染的抗病毒剂
      ≥183 mg/mL
      insoluble in H2O
  7. MLN4924 HCl salt
    A3629 MLN4924 HCl salt
    Target: NAE
    Summary: NAE inhibitor
      Soluble in DMSO
  8. Exendin-4
    A3408 Exendin-4
    中文名: 艾塞那肽
    Target: Glucagon-like peptide 1 (GLP-1) receptors
    Summary: GLP-1激活剂
      ≥145 mg/mL
      ≥52 mg/mL
  9. VX-222 (VCH-222, Lomibuvir)
    A4032 VX-222 (VCH-222, Lomibuvir)
    Target: HCV polymerase
    Summary: HCV RNA聚合酶抑制剂
      ≥44.6 mg/mL
      insoluble in H2O
  10. PSI-6206
    A8189 PSI-6206
     3 Citation
    Target: HCV polymerase
    Summary: HCV RNA聚合酶抑制剂
      ≥13.1 mg/mL
      ≥48.7 mg/mL

10 件产品

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