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Signaling Pathways - 5-alpha Reductases - Mcl-1 - AP-1 - Cytochrome P450 (CYP450)

25件产品中的 11-20

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  1. Thioridazine HCl
    A8537 Thioridazine HCl
    中文名: 盐酸硫利达嗪,盐酸硫代利哒,甲硫达嗪盐酸盐,甲硫哒嗪盐酸盐
    Target: Cytochrome P450 (CYP450)|D1 and D5 Receptors|D2 Receptors|D3 Receptors|D4 Receptors
    Summary: 钙通道蛋白抑制剂
      ≥20.35 mg/mL
      ≥6.78 mg/mL
  2. Posaconazole
    A1718 Posaconazole
    中文名: 泊沙康唑
    Target: Cytochrome P450 (CYP450)|sterol demethylase
    Summary: 甾醇 C14ɑ去甲基化酶抑制剂
      ≥35.04 mg/mL
      insoluble in H2O
  3. Dutasteride
    A1659 Dutasteride
    中文名: 度他雄胺
    Target: 5-alpha Reductases
    Summary: 5-alpha-还原酶抑制剂
      ≥26.43 mg/mL
      ≥13.75 mg/mL
  4. MIM1
    A4465 MIM1
     1 Citation
    Target: Mcl-1
    Summary: Mcl-1抑制剂
      ≥12.15 mg/mL
      insoluble in H2O
  5. Zosuquidar
    A3956 Zosuquidar
    Target: P-glycoprotein (P-gp)|Cytochrome P450 (CYP450)
    Summary: MDR调节剂
      Soluble in DMSO
  6. Dronedarone
    A3374 Dronedarone
    中文名: 决奈达隆
    Target: Cytochrome P450 (CYP450)|sodium channel|adrenergic receptor|potassium channel|calcium channel
    Summary: CYP3A4和2D6抑制剂
      ≥27.84 mg/mL
      insoluble in H2O
  7. Clarithromycin
    A4322 Clarithromycin
    中文名: 克拉霉素
    Target: Cytochrome P450 (CYP450)
    Summary: CYP3A抑制剂
      ≥31.2 mg/mL
      insoluble in H2O
  8. Ketoconazole
    A4316 Ketoconazole
    中文名: 酮康唑
    Target: Cytochrome P450 (CYP450)
    Summary: 环孢菌素氧化酶和睾酮6β-羟化酶的抑制剂
      ≥23.4 mg/mL
      insoluble in H2O
  9. Cobicistat (GS-9350)
    A4313 Cobicistat (GS-9350)
    中文名: 可比司他
    Target: Cytochrome P450 (CYP450)
    Summary: CYP3A的选择性抑制剂
      ≥150.9 mg/mL
      insoluble in H2O
  10. Sabutoclax
    A4199 Sabutoclax
     2 Citation
    Target: Bcl-2|Mcl-1|Bfl-1
    Summary: Pan-Bcl-2抑制剂
      ≥205.6 mg/mL
      insoluble in H2O

25件产品中的 11-20

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