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- B1964 Lonidamine中文名: 氯尼达明Target: HexokinasesSummary: 己糖激酶失活剂
- B2215 Aliskiren Hemifumarate中文名: 阿利克仑半富马酸盐Target: ReninSummary: 肾素抑制剂
- A2571 Pepstatin A1 Citation中文名: 抑肽素Target: Cathepsins|Renin|HIV proteases|PepsinsSummary: 天冬氨酸蛋白酶抑制剂
- A4429 Vialinin ATarget: Deubiquitinating enzymes (DUBs)|IL Receptors|CCL2Summary: USP/IsoT/UCH-L1 DUB抑制剂