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- A4010 Salinosporamide A (NPI-0052, Marizomib)Target: ProteasomeSummary: 20S蛋白酶体抑制剂
- A2571 Pepstatin A1 Citation中文名: 抑肽素Target: Cathepsins|Renin|HIV proteases|PepsinsSummary: 天冬氨酸蛋白酶抑制剂
- A8163 AM 1142 CitationTarget: ProteasomeSummary: 20S蛋白酶体抑制剂
- A2578 Clasto-Lactacystin β-lactoneTarget: ProteasomeSummary: 蛋白酶体抑制剂
- A8179 MG-2621 CitationTarget: ProteasomeSummary: 蛋白酶体抑制剂
- A2604 Celastrol中文名: 雷公藤红素Target: ProteasomeSummary: 抗氧化、抗炎和免疫抑制剂
- B2215 Aliskiren Hemifumarate中文名: 阿利克仑半富马酸盐Target: ReninSummary: 肾素抑制剂
- A8548 Fingolimod (FTY720)中文名: 盐酸芬戈莫德Target: S1P receptorsSummary: S1P受体激动剂
- A4007 MLN97083 Citation中文名: 柠檬酸伊沙佐米Target: ProteasomeSummary: 蛋白酶体抑制剂
- B3225 BAF312 (Siponimod)1 Citation中文名: 辛波莫德Target: S1P receptorsSummary: S1P受体激动剂