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- A2197 Dacarbazine中文名: 达卡巴嗪Target: DNA AlkylatingSummary: 抗肿瘤(恶性黑色素瘤和肉瘤)
- A4383 Tolcapone中文名: 托卡朋Target: Catechol O-Methyltransferase (COMT)Summary: COMT抑制剂
- A4130 ENMD-2076Target: Aurora Kinases|FLT3|RET|Src|VEGFR3/FLT4|NTRK1/TRKA|CSF-1R/c-FmsSummary: Aurora A/Flt3的选择性抑制剂
- A4168 Entacapone中文名: 恩他卡朋Target: Catechol O-Methyltransferase (COMT)Summary: COMT抑制剂
- A2097 Ifosfamide中文名: 异环磷酰胺Target: DNA AlkylatingSummary: 细胞抑制剂