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- A8555 Vandetanib (ZD6474)中文名: 凡德他尼Target: VEGFR|EGFRSummary: VEGFR2/EGFR拮抗剂
- A4118 Hesperadin1 Citation中文名: 橙皮甙,橙皮苷Target: Aurora KinasesSummary: Aurora B抑制剂
- A1926 CA 0742 CitationTarget: CathepsinsSummary: Cathepsin B抑制剂
- A1402 Gemcitabine HCl中文名: 盐酸吉西他滨Summary: 抑制DNA合成,脱氧胞苷类似物
- B5455 G-14 CitationTarget: GPR30Summary: GPR30激动剂
- B7393 GeduninTarget: HSP90Summary: 天然的Hsp90抑制剂
- B7336 Thiostrepton中文名: 硫链丝菌素Target: FoxM1Summary: 抑制细菌蛋白合成的抗生素
- B7157 OGT 2115Target: HeparanasesSummary: 乙酰肝素酶抑制剂
- B6803 Rottlerin1 Citation中文名: 揪毒素Target: PKC|Ca2 /calmodulin-dependent protein kinases (CaMKs)|PRAK|MAPKAP-K2Summary: PKC抑制剂
- B7207 SecinH3Target: Guanine nucleotide exchange factors (GEFs)Summary: Sec7特异性GEF抑制剂