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- A1036 Thrombin Receptor Activator for Peptide 5 (TRAP-5)Target: Thrombin ReceptorSummary: Thrombin Receptor Activator for Peptide 5
- B1012 MS436Target: BromodomainsSummary: BRD4抑制剂
- A4216 Thalidomide中文名: 沙利度胺Target: Ubiquitin E3 LigasesSummary: 免疫调节剂,镇静药,血管生成抑制剂
- B1013 GSK1324726ATarget: BromodomainsSummary: BET蛋白抑制剂
- A4186 Bromosporine1 CitationTarget: BromodomainsSummary: Bromodomain抑制剂
- A4184 PFI-1 (PF-6405761)1 CitationTarget: BromodomainsSummary: BET抑制剂
- B2278 Ibutilide Fumarate中文名: 富马酸伊布利特Target: Voltage-gated Potassium (KV) Channels|Voltage-gated Calcium Channels (CaV)|sodium channelSummary: III类抗心律失常药物
- A3692 OTX-0153 Citation中文名: 比拉瑞塞Target: BromodomainsSummary: BRD抑制剂
- B1989 Nisoldipine中文名: 尼索地平Target: Voltage-gated Calcium Channels (CaV)Summary: 钙通道阻断剂
- A5354 Zonisamide中文名: 唑尼沙胺Target: Voltage-gated Sodium (NaV) Channels|Voltage-gated Calcium Channels (CaV)|Carbonic Anhydrases|Calcium-Activated Potassium (KCa) ChannelsSummary: 抗惊厥和机械效应的抗癫痫药