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- B2161 Nanchangmycin中文名: 南昌霉素Target: AntibioticSummary: 聚醚抗生素
- B3392 GSK269962ATarget: ROCK|RSK|MSKSummary: ROCK抑制剂
- B1293 Y-276329 CitationTarget: ROCKSummary: ROCK选择性抑制剂
- A5611 GSK429286ATarget: ROCKSummary: 选择性ROCK1/ROCK2抑制剂
- A3374 Dronedarone中文名: 决奈达隆Target: Cytochrome P450 (CYP450)|sodium channel|adrenergic receptor|potassium channel|calcium channelSummary: CYP3A4和2D6抑制剂
- B3523 Fasudil中文名: 法舒地尔Target: ROCK|PKC|PKG|PKA|Myosin light chain kinases (MLCKs)Summary: 钙拮抗剂
- B1294 SR-3677Target: ROCKSummary: Rho激酶(ROCK-II)抑制剂
- A4024 Danoprevir (RG7227)中文名: 丹诺瑞韦Target: HCV ProteasesSummary: HCV NS3/4A蛋白酶抑制剂
- B1791 Minocycline HCl中文名: 盐酸米诺环素Target: AntibioticSummary: 四环素抗生素
- A3771 RKI-1447Target: ROCKSummary: ROCK1/ROCK2抑制剂