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- A1036 Thrombin Receptor Activator for Peptide 5 (TRAP-5)Target: Thrombin ReceptorSummary: Thrombin Receptor Activator for Peptide 5
- A3188 ARRY-520 R enantiomerTarget: KspSummary: KSP抑制剂
- A4024 Danoprevir (RG7227)中文名: 丹诺瑞韦Target: HCV ProteasesSummary: HCV NS3/4A蛋白酶抑制剂
- B7675 DIDSTarget: voltage-gated chloride channelsSummary: 阴离子运输抑制剂
- A5343 Ispinesib (SB-715992)中文名: 伊斯平斯Target: KspSummary: 驱动蛋白纺锤体蛋白(KSP)抑制剂