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- A1115 Peptide YY(3-36), PYY, humanTarget: NPY ReceptorsSummary: Y2R激动剂
- B7155 BIBP 3226 trifluoroacetateTarget: NPY Receptors|NPFF receptorSummary: 混合NPY Y1和NPFF受体拮抗剂
- B6552 CGP 20712 dihydrochlorideTarget: adrenoceptorSummary: β1拮抗剂
- B3021 AtglistatinTarget: ATGLSummary: ATGL抑制剂
- A4335 Mildronate中文名: 米屈肼Target: Hydroxylases|carnitine reabsorptionSummary: GBB羟化酶抑制剂
- A8474 Mirabegron (YM178)中文名: 米拉贝隆Target: adrenoceptorSummary: 选择性β3肾上腺素受体激动剂
- A3302 CGI-17461 CitationTarget: BTKSummary: Btk抑制剂