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- B1431 TG003Target: Cdc2-like kinase (Clk)Summary: Cdc2样激酶(Clk)抑制剂
- A4130 ENMD-2076Target: Aurora Kinases|FLT3|RET|Src|VEGFR3/FLT4|NTRK1/TRKA|CSF-1R/c-FmsSummary: Aurora A/Flt3的选择性抑制剂
- A4430 Sivelestat sodium salt中文名: 西维来司钠Target: ElastasesSummary: 白细胞弹性蛋白酶抑制剂
- A4390 Pemetrexed1 Citation中文名: 培美曲塞二钠盐Target: Thymidylate Synthase|DHFR|GARFTSummary: TS、DHFR、GARFT和AICARFT抑制剂