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- A3314 CinaciguatTarget: guanylyl cyclaseSummary: 可溶性鸟苷酸环化酶(sGC)激活剂
- A8660 Cilengitide1 Citation中文名: 西仑吉肽Target: IntegrinsSummary: 整合素αvβ3和αvβ5的抑制剂
- B1685 Broxyquinoline中文名: 溴羟喹啉Target: Tetrahydrofolate dehydrogenaseSummary: 抗原虫剂
- A8601 Tankyrase Inhibitors (TNKS) 49Target: TankyrasesSummary: 端锚聚合酶抑制剂