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- A8610 6,2',4'-TrimethoxyflavoneTarget: Aryl hydrocarbon receptors (AHRs)Summary: 芳基烃受体拮抗剂
- A4125 CYC116Target: Aurora Kinases|FLT3|VEGFRSummary: Aurora A/B抑制剂
- A1912 Lomeguatrib中文名: 罗米鲁曲Target: O6-methylguanine-DNA-methyl-transferase (MGMT)Summary: MGMT抑制剂
- A3408 Exendin-4中文名: 艾塞那肽Target: Glucagon-like peptide 1 (GLP-1) receptorsSummary: GLP-1激活剂
- A3847 SU5416中文名: 司马沙尼Target: VEGFRSummary: VEGF受体抑制剂和AHR激动剂
- A8313 RAF265Target: Raf|VEGFRSummary: 多细胞激酶抑制剂