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- A3278 Nonivamide (Capsaicin Analog)1 Citation中文名: 香草壬酰胺Target: TRP ChannelSummary: TRPV1受体激动剂
- A3850 TAK-2427 Citation中文名: 瑞沙托维Target: Toll-like receptors (TLRs)|NO Donors / Precursors|IL ReceptorsSummary: TLR 4信号抑制剂
- A4329 Cilomilast中文名: 西洛司特Target: Phosphodiesterases (PDEs)Summary: PDE4抑制剂
- A4317 Apremilast (CC-10004)中文名: 阿普斯特Target: Phosphodiesterases (PDEs)Summary: PDE4抑制剂
- A1907 5-Azacytidine6 Citation中文名: 氮胞苷(5-氮胞苷)Target: DNA MethyltransferasesSummary: DNA甲基转移酶抑制剂