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- A8651 LY2940680Target: Smoothened receptorSummary: Hedgehog / SMO拮抗剂,抑制Hh信号。
- A4483 PRIMA-1Target: p53Summary: BAX抑制剂
- A4390 Pemetrexed1 Citation中文名: 培美曲塞二钠盐Target: Thymidylate Synthase|DHFR|GARFTSummary: TS、DHFR、GARFT和AICARFT抑制剂
- A4203 Tenovin-1Target: Sir2-like Family Deacetylases (Sirtuins)|p53|p21Summary: SIRT2 抑制剂,p53激活剂