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- A2278 NVP-AEW541Target: Insulin ReceptorSummary: IGF-IR抑制剂
- A8528 TAK-285Target: EGFR|HER2Summary: HER2/EGFR(HER1)抑制剂
- B2172 PP121Target: mTOR|Eph Receptors|VEGFR|PDGFR|Bcr-Abl|Src|DNA-PK|P110|HckSummary: 酪氨酸激酶和磷酸肌醇激酶双重抑制剂
- N1659 1-Deoxynojirimycin中文名: 1-脱氧野尻霉素Target: GlucosidasesSummary: anti-cancer medicine