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- A1185 BMS-754807Target: Insulin and Insulin-like ReceptorsSummary: 有效的、选择性的IGF-1R和InsR抑制剂
- A8440 GSK1838705ATarget: Insulin and Insulin-like Receptors|ALKSummary: ATP竞争性IGF-IR/IR/ALK抑制剂
- A1302 GSK1904529ATarget: Insulin and Insulin-like ReceptorsSummary: IGF-1R/IR 选择性抑制剂
- B4357 UNC2881Target: Mer tyrosine kinaseSummary: Mer酪氨酸激酶抑制剂
- B3209 TriapineTarget: Ribonucleotide ReductasesSummary: 核糖核苷酸还原酶(ribonucleotide reductase)抑制剂