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- A4390 Pemetrexed1 Citation中文名: 培美曲塞二钠盐Target: Thymidylate Synthase|DHFR|GARFTSummary: TS、DHFR、GARFT和AICARFT抑制剂
- A2597 Brivanib (BMS-540215)中文名: 布立尼布Target: VEGFR|FGFR|Flk1Summary: VEGFR-2的ATP竞争性抑制剂
- B3709 Midostaurin (PKC412)中文名: 米哚妥林Target: PKC|PKA|KDR|Flk1|PPK|c-Syk|CDK1/CyclinBSummary: PKC抑制剂
- B6787 STO-609 acetateTarget: CaM-KKSummary: Ca2+-钙调蛋白依赖性蛋白激酶激酶抑制剂
- A8633 Concanamycin A1 Citation中文名: 卡那霉素ATarget: Vacuolar-type ATPaseSummary: V型(液泡)H +-ATP酶抑制剂