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- A3220 Bardoxolone中文名: 巴多索隆Target: COX|iNOSSummary: 用于治疗慢性肾病,每天一次
- A3023 P0050911 CitationTarget: Ubiquitin-specific proteasesSummary: 泛素特异性蛋白酶7(USP7)抑制剂
- B1964 Lonidamine中文名: 氯尼达明Target: HexokinasesSummary: 己糖激酶失活剂
- B5839 SU6656Target: Src|Lyn|YES|FynSummary: Src 酪氨酸激酶抑制剂
- A4124 TAK-901Target: Aurora Kinases|FLT3|Src|JAK|LRRK2|Hck|FGR|YES|Fyn|ARGSummary: Aurora A/B抑制剂