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- A8366 ARRY-380Target: HER2Summary: 酪氨酸激酶HER2和P95-HER2抑制剂。
- B5839 SU6656Target: Src|Lyn|YES|FynSummary: Src 酪氨酸激酶抑制剂
- A4383 Tolcapone中文名: 托卡朋Target: Catechol O-Methyltransferase (COMT)Summary: COMT抑制剂
- A2942 Masitinib (AB1010)中文名: 马赛替尼Target: PDGFR|c-Kit|LynSummary: 酪氨酸激酶抑制剂
- A4168 Entacapone中文名: 恩他卡朋Target: Catechol O-Methyltransferase (COMT)Summary: COMT抑制剂
- A5354 Zonisamide中文名: 唑尼沙胺Target: Voltage-gated Sodium (NaV) Channels|Voltage-gated Calcium Channels (CaV)|Carbonic Anhydrases|Calcium-Activated Potassium (KCa) ChannelsSummary: 抗惊厥和机械效应的抗癫痫药
- A4364 Methazolamide中文名: 醋甲唑胺Target: Carbonic AnhydrasesSummary: 碳酸酐酶抑制剂
- B1279 Dorzolamide中文名: 多佐胺Target: Carbonic AnhydrasesSummary: 碳酸酐酶抑制剂
- A8408 Dichlorphenamide中文名: 双氯非那胺Target: Carbonic AnhydrasesSummary: 碳酸酐酶抑制剂
- A3145 Afatinib dimaleate中文名: 马来酸阿法替尼Target: EGFR|HER2Summary: EGFR抑制剂