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- N1336 Chrysin中文名: 柯因,5,7-二羟黄酮Target: Estrogen and Related Receptors|Hypoxia Inducible Factors (HIFs)Summary: 抗炎和抗肿瘤试剂
- B1518 Erteberel (LY500307)Target: Estrogen and Related ReceptorsSummary: ERβ激动剂
- B4658 LY451395Target: AMPASummary: 变构调节剂
- A8425 Estradiol中文名: 雌二醇Target: Estrogen and Related ReceptorsSummary: 性激素
- B6004 PX-478 2HClTarget: Hypoxia Inducible Factors (HIFs)Summary: HIF-1α抑制剂
- A8534 Terfenadine中文名: 特非那定Target: Voltage-gated Potassium (KV) Channels|Histamine H1 Receptors|Inward Rectifier Potassium (Kir) ChannelsSummary: 组胺H1受体拮抗剂
- B1198 CisaprideTarget: Voltage-gated Potassium (KV) Channels|5-HT4 ReceptorSummary: 5-HT4受体激动剂
- B1506 Estradiol valerate中文名: 戊酸雌二醇Target: Estrogen and Related ReceptorsSummary: 雌激素受体激动剂
- B1115 BAY 87-2243Target: Hypoxia Inducible Factors (HIFs)Summary: 有效的HIF-1选择性抑制剂
- B1513 Toremifene Citrate中文名: 枸橼酸托瑞米芬Target: Estrogen and Related ReceptorsSummary: 口服选择性雌激素受体调节剂(SERM)