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- N2135 Gossypol2 Citation中文名: 棉籽酚,棉酚Target: DehydrogenaseSummary: PAF抑制剂,抗生育和抗癌
- A3302 CGI-17461 CitationTarget: BTKSummary: Btk抑制剂
- A4182 Resveratrol2 Citation中文名: 白藜芦醇Target: Sir2-like Family Deacetylases (Sirtuins)|COX|LOX|Adenylyl cyclase|Quinone reductaseSummary: SIRT1激活剂
- B5986 Enoxolone中文名: 甘草次酸Target: DehydrogenaseSummary: 甘草的主要成分
- B6185 ACP-196中文名: 阿卡替尼Target: BTKSummary: 不可逆的BTK抑制剂