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- A8366 ARRY-380Target: HER2Summary: 酪氨酸激酶HER2和P95-HER2抑制剂。
- B7785 LDN 209929 dihydrochlorideTarget: haspin kinaseSummary: Haspin激酶抑制剂
- B1463 KPT-276Target: nuclear export|CRM1Summary: CRM1抑制剂
- A3145 Afatinib dimaleate中文名: 马来酸阿法替尼Target: EGFR|HER2Summary: EGFR抑制剂
- A8528 TAK-285Target: EGFR|HER2Summary: HER2/EGFR(HER1)抑制剂