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- A3237 Betulinic acid中文名: 白桦脂酸,桦木酸Target: Aminopeptidases|Topoisomerases|HIVSummary: 抗HIV和抗肿瘤化合物,五环三萜类化合物
- A8644 Acyclovir中文名: 阿昔洛韦Target: HSVSummary: 抗病毒剂
- B4745 (S)-10-Hydroxycamptothecin中文名: 羟喜树碱Target: TopoisomerasesSummary: 拓扑异构酶I抑制剂
- B1029 BAY 57-1293中文名: 普瑞利韦Target: HSVSummary: HSV解旋酶-引物酶抑制剂
- B1809 Penciclovir中文名: 喷昔洛韦Target: HSVSummary: HSV-1 DNA合成抑制剂
- A8400 Clinafloxacin CI96 AM1091中文名: 克林沙星Target: TopoisomerasesSummary: 拓扑异构酶抑制剂
- A2601 Aclacinomycin ATarget: TopoisomerasesSummary: 拓扑异构酶I和II的双重抑制剂
- N2133 7-Ethyl-10-hydroxycamptothecinTarget: TopoisomerasesSummary: TOPO I抑制剂
- A5511 Ofloxacin中文名: 氧氟沙星Target: Topoisomerases|DNA gyraseSummary: 氟喹诺酮类抗生素
- B2295 Pirarubicin1 Citation中文名: 吡柔比星Target: TopoisomerasesSummary: 拓扑异构酶II抑制剂,蒽环类抗生素