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- A8229 ML161Target: Protease-Activated ReceptorsSummary: PAR1抑制剂
- A2198 Genistein中文名: 金雀异黄酮,染料木素Target: Estrogen and Related Receptors|PPAR|PTKSummary: ER agonist
- A8809 Vorapaxar中文名: 沃拉帕沙Target: Protease-Activated ReceptorsSummary: PAR-1拮抗剂
- A2689 Butein中文名: 紫铆因,紫铆查尔酮Target: Src|STAT|EGFR|Angiotensin-Converting Enzymes (ACEs)|5-Lipoxygenases|PTK|enoyl-acyl-carrier protein reductaseSummary: 蛋白激酶抑制剂
- N1308 Biochanin A中文名: 鹰嘴豆芽素A,鸡豆黄素ATarget: EGFR|FAAH|PTKSummary: 脂肪酸酰胺水解酶的天然抑制剂
- A4130 ENMD-2076Target: Aurora Kinases|FLT3|RET|Src|VEGFR3/FLT4|NTRK1/TRKA|CSF-1R/c-FmsSummary: Aurora A/Flt3的选择性抑制剂