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- A4010 Salinosporamide A (NPI-0052, Marizomib)Target: ProteasomeSummary: 20S蛋白酶体抑制剂
- A8204 Lopinavir中文名: 洛匹那韦Summary: HIV蛋白酶抑制剂
- A4005 RO49290971 CitationSummary: γ-secretase抑制剂
- A4056 AT13387Target: HSP90Summary: Hsp90抑制剂
- A4015 Disulfiram中文名: 双硫仑Target: Aldehyde DehydrogenasesSummary: 多巴胺β-羟化酶抑制剂
- B2127 Rifapentine中文名: 利福喷丁Target: RNA PolymerasesSummary: 治疗肺结核的抗生素药物.
- A3859 Tariquidar methanesulfonate, hydrate中文名: 他立喹达二甲磺酸盐六水合物Target: P-glycoprotein (P-gp)Summary: P-糖蛋白抑制剂
- A8208 Tariquidar2 Citation中文名: 他立喹达Target: P-glycoprotein (P-gp)Summary: P-糖蛋白抑制剂
- A3018 Trametinib (GSK1120212)7 Citation中文名: 曲美替尼Target: MEKSummary: MEK1和MEK2抑制剂
- A3021 GDC-0449 (Vismodegib)1 Citation中文名: 维莫德吉Target: P-glycoprotein (P-gp)|HedgehogSummary: Hedgehog拮抗剂