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- A2602 Calpain Inhibitor I, ALLN2 CitationTarget: Cathepsins|CalpainsSummary: Calpain I/II/ B/L抑制剂
- A4413 PD 150606Target: CalpainsSummary: 非肽类钙蛋白酶抑制剂
- A2451 Epirubicin HCl中文名: 盐酸表阿霉素Target: TopoisomerasesSummary: 抗生素类抗肿瘤药物
- A3237 Betulinic acid中文名: 白桦脂酸,桦木酸Target: Aminopeptidases|Topoisomerases|HIVSummary: 抗HIV和抗肿瘤化合物,五环三萜类化合物
- A5511 Ofloxacin中文名: 氧氟沙星Target: Topoisomerases|DNA gyraseSummary: 氟喹诺酮类抗生素
- P10019 Prulifloxacin (Pruvel)中文名: 普鲁利沙星Target: Topoisomerases
- B4745 (S)-10-Hydroxycamptothecin中文名: 羟喜树碱Target: TopoisomerasesSummary: 拓扑异构酶I抑制剂
- A3381 Edoxaban中文名: 依度沙班Target: Factor XaSummary: 因子Xa抑制剂
- A3126 5-R-Rivaroxaban中文名: 5-R-利伐沙班Target: Factor XaSummary: 因子Xa(FXa)抑制剂
- A1971 Etoposide4 Citation中文名: 依托泊苷Target: TopoisomerasesSummary: 拓扑异构酶II(Topo II)抑制剂