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- A8182 3-Deazaneplanocin A (DZNep) hydrochloride1 Citation中文名: 3-去氮腺嘌呤A盐酸盐Target: EZH2Summary: SAHH和EZH2抑制剂
- A3196 AT-101中文名: (R)-(-)-棉子酚Target: NS3/4a ProteasesSummary: BH3-类似物,棉酚对映异构体
- A5618 Daclatasvir (BMS-790052)中文名: 达卡他韦Target: HCV ProteasesSummary: HCV NS5A抑制剂
- B1474 FT-207 (NSC 148958)中文名: 替加氟Summary: DNA/RNA合成抑制剂
- B1858 Tranexamic Acid中文名: 氨甲环酸Target: fibrinolysisSummary: 纤溶酶原激活的竞争性抑制剂
- A3014 BGJ3981 CitationTarget: FGFRSummary: FGFR抑制剂