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- B5624 STF 083010Target: Inositol-requiring enzyme 1 (IRE1)Summary: IRE1α核酸内切酶抑制剂
- B6429 Naltrindole hydrochloride中文名: 纳曲吲哚盐酸盐Summary: δ阿片样物质拮抗剂
- B5638 ACHPSummary: IκB激酶抑制剂
- A4093 ITF2357 (Givinostat)2 CitationTarget: Histone Deacetylases (HDACs)Summary: HDAC抑制剂
- A2168 Dovitinib (TKI-258, CHIR-258)2 Citation中文名: 多韦替尼Target: FLT3|VEGFR|PDGFR|c-Kit|FGFRSummary: 多靶点RTK抑制剂
- A3692 OTX-0153 Citation中文名: 比拉瑞塞Target: BromodomainsSummary: BRD抑制剂