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- A4024 Danoprevir (RG7227)中文名: 丹诺瑞韦Target: HCV ProteasesSummary: HCV NS3/4A蛋白酶抑制剂
- A2224 Stattic5 CitationTarget: STATSummary: STAT3抑制剂
- B1879 AdipoRonTarget: AdipoR1|AdipoR2Summary: AdipoR1/2激动剂
- A4416 AZ 10417808Target: CaspasesSummary: Caspase-3抑制剂
- B1472 Mizoribine中文名: 咪唑立宾Target: Synthases/SynthetasesSummary: DNA/RNA合成抑制剂
- A3368 DMAT2 CitationTarget: Pim|CK2|HIPK2|HIPK3Summary: CK2抑制剂
- A8637 IOWH-032Target: CFTRSummary: CFTR抑制剂
- B1087 GlyH-101Target: CFTRSummary: CFTR Inhibitor II
- A8300 ZCL2781 CitationTarget: Cdc42Summary: Cdc42抑制剂
- B1307 SJB3-019ATarget: USPSummary: Usp1抑制剂