Leukotriene Receptor
Leukotrienes receptors are divided into two types, BLT receptors and CycLT receptors. BLT receptors mediate chemoattraction. CysLT receptors mediate pro-inflammatory effects including constriction of airways ad smooth muscle contraction.
- C5518 γ-Linolenic Acid中文名: γ-亚麻酸Summary: 弱LTB4受体拮抗剂
- C5416 REV 5901Summary: 半胱氨酰-白三烯受体的拮抗剂
- C5226 γ-Linolenic Acid methyl esterSummary: 弱白三烯B4(LTB4)受体拮抗剂
- C4677 LY223982Summary: 有效的BLT1受体拮抗剂
- C4837 5(S),6(R)-7-trihydroxymethyl HeptanoateSummary: 抑制白三烯B4(LTB4)诱导的多形核嗜中性粒细胞(PMN)趋化性
- C4323 ARM1Summary: LTB4合成抑制剂
- C3082 HAMI3379Summary: CysLT2受体拮抗剂
- C3110 LY171883Summary: 白三烯D4受体拮抗剂,口服有效
- B8031 MK-571 sodium salt hydrate3 CitationTarget: CysLT1Summary: CysLT1受体拮抗剂
- B6978 LY 255283Summary: BLT2受体拮抗剂