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Signaling Pathways - GABAB Receptors - Histamine H2 Receptors - Angiotensin AT1 Receptors - sodium channel

10 件产品

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  1. CGP 55845 hydrochloride
    B5086 CGP 55845 hydrochloride
    Target: GABAB Receptors
    Summary: GABAB受体拮抗剂
      <43.87 mg/mL
  2. Ranitidine
    B1564 Ranitidine
    中文名: 盐酸雷尼替丁
    Target: Histamine H2 Receptors
    Summary: 组胺H2受体拮抗剂
      ≥17.54 mg/mL
      ≥99 mg/mL
  3. Ibutilide Fumarate
    B2278 Ibutilide Fumarate
    中文名: 富马酸伊布利特
    Target: Voltage-gated Potassium (KV) Channels|Voltage-gated Calcium Channels (CaV)|sodium channel
    Summary: III类抗心律失常药物
      ≥25.6 mg/mL
      ≥16.4 mg/mL
  4. Lamotrigine
    B2249 Lamotrigine
     1 Citation
    中文名: 拉莫三嗪
    Target: 5-HT receptors|sodium channel
    Summary: 5-HT抑制剂,钠通道阻断剂
      ≥12.3 mg/mL
      insoluble in H2O
  5. Valsartan
    B2214 Valsartan
    中文名: 缬沙坦
    Target: Angiotensin AT1 Receptors
    Summary: 血管紧张素II AT1受体拮抗剂
      ≥19.65 mg/mL
      insoluble in H2O
  6. (R)-baclofen
    B1531 (R)-baclofen
    中文名: (R)-巴氯芬
    Target: GABAB Receptors
    Summary: GABA受体激动剂
      insoluble in DMSO
      ≥7.13 mg/mL
  7. AVE 0991
    B1007 AVE 0991
     1 Citation
    Target: Angiotensin AT1 Receptors
    Summary: 血管紧张素-(1-7)受体激动剂
      ≥29.04 mg/mL
  8. Azilsartan
    B2210 Azilsartan
    中文名: 阿齐沙坦
    Target: Angiotensin AT1 Receptors
    Summary: 强效血管紧张素II 1型(AT1)受体反向激动剂
      ≥16.95 mg/mL
      insoluble in H2O
  9. Irbesartan
    A5970 Irbesartan
    中文名: 安博维,厄贝沙坦
    Target: Angiotensin AT1 Receptors
    Summary: 血管紧张素II抑制剂
      ≥17.4 mg/mL
      insoluble in H2O
  10. Dronedarone
    A3374 Dronedarone
    中文名: 决奈达隆
    Target: Cytochrome P450 (CYP450)|sodium channel|adrenergic receptor|potassium channel|calcium channel
    Summary: CYP3A4和2D6抑制剂
      ≥27.84 mg/mL
      insoluble in H2O

10 件产品

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